Other Janus Kinase Inhibitors

JAK inhibitor Route Target Current clinical trials or reported use
Delgocitinib Topical Pan-JAK Atopic dermatitis, discoid lupus, chronic hand eczema
Cerdulatinib Topical Pan-JAK, SYK Vitiligo
Gusacitinib Oral Pan-JAK, SYK Atopic dermatitis
Peficitinib Oral Pan-JAK Psoriasis
Beprocitinib Oral JAK1/TK2 Alopecia areata; atopic dermatitis; hidradenitis suppurativa; plaque psoriasis; psoriatic arthritis, vitiligo
Itacitinib Oral JAK-1,2 Psoriasis, melanoma, chronic itch
Filgotinib Oral JAK1 Cutaneous lupus
Lestaurtinib Oral JAK2 Psoriasis
Deucravacitinib Oral Regulatory domain of TYK2 Psoriasis.
Note: initial studies showed no laboratory abnormalities, as seen with other JAK inhibitors
Ritlecitinib Oral JAK3/TEC Alopecia areata (phase III), vitiligo (phase II)